Indications

lead translational priority-epigenetic bone regeneration

Development Opportunities

•Known/prototype compounds
Commercially available candidates with preclinical support
Example: GSK126, tazemetostat
•Extensor lead compounds
First in class nuclear bone stimulators (EBI-700 series)
Prior SBIR/R43-supported development foundation
•Novel Extensor-Cayman collaboration compounds
New chemical matter with stronger material IP potential
Current translational priority

SECONDARY AREAS OF INVESTIGATION

Osteoarthritis

Novel approaches to degeneration and joint preservation.

Fibrosis

Targeting pathological soft tissue remodeling and fibrosis.

Inflammatory Musculoskeletal Disease

Exploring pathways involved in chronic musculoskeletal inflammation and tissue dysfunction.